I-Drotaverine Hydrochloride noma amaphilisi e-Drotaverine HCL ayimithi yomlomo esetshenziselwa izinhlungu kanye namajaqamba ngenxa yokuphuma emathunjini, ukuya esikhathini, noma ngezinye izikhathi ubuhlungu bokubeletha. Nakuba kusebenza, umuntu ohlushwa yinoma ibuphi izinhlungu noma izinhlungu akumele abe nalo muthi ngaphandle kwemvume kadokotela, njengoba kungase kubangele umonakalo omkhulu noma imiphumela engemihle.
I-Drotaverine Hydrochloride, eyaziwa nangokuthi i-drotaverine, iyisidakamizwa se-antispasmodic. Isebenza ngempumelelo ekwelapheni ama-spasms noma ama-twitches emisipha ebushelelezi yamathumbu, kanye nobuhlungu obubangelwa i-bowel syndrome ecasulayo, bekhanda, ubuhlungu bokuya esikhathini noma ama-cramps, izinhlungu zomlomo wesibeletho ngesikhathi sokubeletha, njll. Ihlobene ngokwesakhiwo ne-papaverine kodwa ikhombisa amandla amakhulu kune-papaverine.
I-Drotaverine Hydrochloride iyithebhulethi ye-antispasmodic esetshenziselwa ukukhulula ama-spasms namajaqamba, njengobuhlungu bokuya esikhathini, isisu ubuhlungu, ubuhlungu besifuba, ubuhlungu ngenxa izinso namatshe e-biliary, nobuhlungu besisu. Ngaphezu kwalokho, i-Drotaverine Hydrochloride iphatha ngokuyinhloko ukufinyela kwemisipha ebushelelezi, okuzwakala njengobuhlungu besisu obuphindaphindiwe emgudwini wamathumbu. Iphinde ikhulule ubuhlungu ngenxa ye-bowel syndrome ecasulayo kanye ne-spasms yomlomo wesibeletho.
I-Atropine, i-diclofenac, i-levodopa, ne-diazepam ingeminye yemithi engase ihlangane ne-Drotaverine Hydrochloride. Ngakho-ke, kuyatuseka ukufuna usizo lwezokwelapha ngaphambi kokusebenzisa umuthi.
Imiphumela emibi ye-Drotaverine Hydrochloride ayivamile. Noma kunjalo, nazi ezinye zezimpawu isiguli esingase sibe nazo:
Kubalulekile ukubika kudokotela uma kukhona imiphumela engemihle, njengoba kushiwo ngenhla, noma yimiphi imiphumela emibi emisha. Udokotela angase ashintshe umuthi noma aguqule umthamo womuthi.
Kunconywa ukuthatha amaphilisi e-Drotaverine HCL ngokweseluleko sikadokotela. Nokho, nansi eminye yemithamo enconyiwe:
Ukukhuluma nodokotela ngaphambi kokuthatha i-Drotaverine Hydrochloride kubalulekile, ikakhulukazi uma ungezwani nemithi ethile ngenxa yezithako ezithile ezisebenzayo. Akumele kuthathwe ngemithamo emikhulu kodwa ngengilazi egcwele amanzi. Futhi, uma kwenzeka kuba nemiphumela engemihle, kubalulekile ukubonana nodokotela. Ngaphezu kwalokho, funa usizo lwezokwelapha uma izimpawu zingathuthuki, futhi khumbula ukungawusebenzisi umuthi ngemva kokuphelelwa yisikhathi.
Ukusetshenziswa kwe-drotaverine ephumuza imisipha ebushelelezi ngesikhathi sokukhulelwa kungase kube yingozi, ikakhulukazi phakathi ne-trimester yokuqala. Ezinye izinto ezingasebenzi emkhiqizweni zingase zibangele ukungezwani okukhulu noma ezinye izinkinga. Kungalimaza umama noma kuphazamise ukukhula kombungu. Ngakho, ukuze kuhlolwe isilinganiso sengozi nenzuzo nokukhetha inkambo ephephe kunazo zonke, odokotela kufanele babe nalolu lwazi.
Uma kwenzeka uphuthelwe umthamo, phuza umuthi ngokushesha nje lapho ukhumbula. Kodwa-ke, uma umthamo olandelayo useduze, ungase ufune ukulinda umthamo olandelayo futhi ungathathi umuthi owengeziwe ukuze uvale imithamo egejiwe. Khumbula ukuthi ungaphuthelwa yinoma yimuphi umthamo ukuze uqinisekise ukusebenza kahle kwawo.
Esimeni se-overdose, funa usizo lwezokwelapha ngokushesha uma uqala ukuzizwa unesiyezi, ukozela, nokungahlaliseki noma ukushaya kwenhliziyo okwedlulele. Ubukhulu bezimpawu bungahluka, kodwa kubalulekile ukukhuluma nodokotela ngakho.
Gcina isitsha somuthi sivalwe ngokuqinile endaweni eyomile futhi enomoya omuhle. Ungawubeki elangeni; uyibeke endaweni ephakeme lapho izingane zingakwazi ukufinyelela kuyo.
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I-Drotaverine Hydrochloride |
I-Dicyclomine |
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I-Drotaverine Hydrochloride iyimithi ye-antispasmodic efana ne-papaverine ngesakhiwo, futhi ayinazo izakhiwo ze-anticholinergic. |
Ithebhulethi ye-Dicyclomine umuthi kadokotela otholakala ngaphansi kwegama lomkhiqizo we-Bentyl. |
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Ivimbela i-PDE4 enzyme (ikhulula imisipha) |
Ivimbela i-acetylcholine (ikhulula imisipha) |
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Amathebulethi, Amaphilisi, Imijovo (kwamanye amazwe) |
Amathebulethi, Amaphilisi, Imijovo (kwamanye amazwe) |
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Isisu/Amajaqamba emathunjini, Biliary colic |
Amajaqamba e-IBS, izilonda zesisu, i-Diverticulitis |
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Ikhanda elibuhlungu, Isicanucanu, Ukuqunjelwa |
Umlomo owomile, ukungaboni kahle, isiyezi, ukozela, ukuqunjelwa (nokudideka kubantu abadala) |
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I-OTC (amazwe amaningi), Incwadi kadokotela (amanye) |
Incwadi kadokotela kuphela |
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Ukusebenzisana okungenzeka, thintana nodokotela |
Ukusebenzisana okungenzeka, thintana nodokotela |
I-Drotaverine Hydrochloride ikhulula imisipha ebushelelezi, ngokuyinhloko iqondise isisu kanye namajaqamba emathunjini noma i-biliary colic. Ngokujwayelekile ukubekezelelwa kahle, kungabangela ubuhlungu bekhanda, isicanucanu, kanye nokuqunjelwa. Nakuba itholakala ezitolo emazweni amaningi, kungcono ukubonana nodokotela ngaphambi kokuyisebenzisa ukuze uqinisekise ukuthi ikulungele futhi uxoxe ngemiphumela engemihle engaba khona nokusebenzisana.
Izimpendulo. Ukuphepha kwe-Drotaverine Hydrochloride akukakasungulwa. Ngokusho kwe-FDA (Food and Drug Administration) yase-USA, i-Drotaverine Hydrochloride ihlukaniswa njengengaba yingozi. Ngakho-ke, kufanele isetshenziswe kuphela lapho izinzuzo zidlula ubungozi bayo. Umuthi unikezwa ukunciphisa ama-spasms we-gastrointestinal kanye ne-genitourinary muscle ngesikhathi ukukhulelwa.
Izimpendulo. I-Drotaverine Hydrochloride ingathathwa ngenxa yobuhlungu besisu, njengoba umphumela we-antispasmodic we-Drotaverine Hydrochloride ubonisa umphumela ophumuzayo ngendlela emangalisayo emisipha ebushelelezi yamathumbu, esiza ekudambiseni ubuhlungu ngaphandle kwemiphumela emibi ye-anticholinergic.
Izimpendulo. I-Drotaverine Hydrochloride ne-paracetamol ingathathwa ndawonye. Nokho, ukukhuluma nodokotela ngaphambi kokuhlanganisa le mithi emibili kuyancomeka. Ukuzelapha ngenkathi uhlanganisa lezi ezimbili akuvunyelwe ngokuphelele. Lokhu kungenxa yokuthi ukusebenzelana kungase kube nomthelela we-synergistic.
Izimpendulo. Amaphilisi e-Drotaverine HCL angamaphilisi ezinhlungu futhi asebenza kahle kakhulu esimweni sobuhlungu obuvela emisipha ebushelelezi. I-Drotaverine hydrochloride iyi-antispasmodic engakwazi ukukhulula futhi inciphise ama-spasms nama-cramps angase avele ngenxa yemisipha ebushelelezi.
Izimpendulo. Cha, i-Drotaverine Hydrochloride ayiwona ama-antibiotic. I-Drotaverine Hydrochloride iyisidakamizwa se-antispasmodic esivimbela i-PDE4. Ngakho-ke, ukugwema ukuboshwa kwe-cAMP ku-PDE4 kubangela ukuxegiswa kwemisipha ebushelelezi. Ngakho-ke, ayikwazi ukumisa noma yiziphi izifo.
Izimpendulo. I-Drotaverine Hydrochloride ngokuvamile ithatha imizuzu engu-20-30 ukuze isebenze ngemva kokuyithatha.