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I-Pregabalin

I-Pregabalin imithi enamandla eyingxenye yezidakamizwa ezibizwa ngokuthi ama-anticonvulsants. Lesi sidakamizwa esisebenziseka ngezindlela eziningi siye saqashelwa ngekhono laso lokubhekana nezimo ezihlukahlukene zezokwelapha. I-Pregabalin inethonya ohlelweni lwezinzwa ngokuthulisa izinzwa ezisebenza ngokweqile emzimbeni. Ukwakheka kwayo kufana ne-gamma-aminobutyric acid (GABA), i-neurotransmitter evimbela ebuchosheni. 

Ukusetshenziswa kwethebhulethi ye-Pregabalin

I-Pregabalin inqunyelwe ukwelapha izimo zezokwelapha ezahlukahlukene. Umsebenzi wawo oyinhloko ukuthulisa izinzwa ezisebenza ngokweqile emzimbeni, okuwenza uphumelele ekulawuleni izinhlobo eziningana zobuhlungu nokuphazamiseka kwezinzwa, okuhlanganisa:

  • Amaphilisi e-Pregabalin anokusetshenziswa okubalulekile ekudambiseni ubuhlungu be-neuropathic, obubangelwa yimizwa elimele. 
  • Okunye ukusetshenziswa kwe-pregabalin okubalulekile ekwelapheni i-postherpetic neuralgia. Lesi simo sibangela ukuvutha, ukugwazwa ubuhlungu noma izinhlungu ezingase ziqhubeke izinyanga noma ngisho neminyaka ngemva kokuba a shingles ukuphuma. 
  • Ama-capsules we-Pregabalin nesisombululo somlomo anokusetshenziswa ekwelapheni i-fibromyalgia, isimo esihlala isikhathi eside esibonakala ngokuqina kwemisipha nokuzwela, ubuhlungu, ukukhathala, nobunzima bokulala noma ukulala..
  • I-Pregabalin iphinde ibe nokusetshenziswa ekudambiseni ubuhlungu be-neuropathic obungenzeka ngemva kokulimala komgogodla. 
  • Ama-capsules we-Pregabalin kanye nezixazululo zomlomo nazo ziyasebenza ekwelapheni okuthile izinhlobo zokuquleka kokubili abadala kanye nezingane. 

Ungayisebenzisa kanjani i-Pregabalin Tablet

I-Pregabalin iza ngezindlela ezihlukahlukene namandla ukuze ivumelane nezidingo zezokwelapha ezihlukene. Kubalulekile ukuthi uphuze lo muthi njengoba nje udokotela esho. 

Lapho uthatha i-pregabalin, iziguli kufanele zilandele le mihlahlandlela:

  • Thatha umuthi ngesikhathi esifanayo nsuku zonke ukuze ugcine amazinga angaguquki emzimbeni.
  • Ungathatha i-pregabalin capsule noma uketshezi lomlomo ngokudla noma ngaphandle kokudla.
  • Ukuze uthole amaphilisi akhishwe isikhathi eside, waphuze ngemva kokudla kwakusihlwa. Igwinye ithebhulethi iphelele ngaphandle kokuyiphula noma ukuyihlafuna.
  • Uma usebenzisa uketshezi lomlomo, lukale ngokunembile usebenzisa isipuni sokulinganisa esimakiwe noma inkomishi yokwelapha. 

Imiphumela Emibi ye-Pregabalin Tablet

  • Isiyezi kanye nobuthongo
  • Umbono ophundlekile
  • Umlomo omile
  • Inzuzo yesisindo
  • I-nausea nokuhlanza
  • Ukubunzima ukugxila
  • Ukwenyuka kwesifiso sokudla (ikakhulukazi ezinganeni)
  • Kulabo abathatha amaphilisi akhishwa isikhathi eside, ubuhlungu bekhanda, ukukhathala, nesicanucanu nakho kuvamile.
  • Ezimweni ezimbi kakhulu, i-pregabalin ingase ibangele ukungezwani komzimba - ukuqubuka kwesikhumba, ukulunywa, ukuqubuka, ukuvuvukala kobuso, amehlo, izindebe, ulimi, izingalo, noma imilenze, nokuphefumula kanzima.

Ukuqapha

I-Pregabalin, nakuba isebenza ezimweni ezihlukahlukene, idinga ukucatshangelwa nokuqapha ngokucophelela: 

  • Iziguli akufanele zisebenzise lo muthi uma zine-allergies kuwo.
  • Kubalulekile ukwazisa udokotela nganoma yiziphi izimo esezivele zikhona, okuhlanganisa izifo zamaphaphu ezifana nesifo esingamahlalakhona sokuvimbela i-pulmonary (COPD), ukuphazamiseka kwemizwelo, izinkinga zenhliziyo (ikakhulukazi ukwehluleka kwenhliziyo eqinile), ukuphazamiseka kwegazi, isifo sezinso, isifo sikashukela, ukuba umlutha wezidakamizwa noma utshwala, noma umlando wokungezwani okukhulu komzimba.
  • I-Pregabalin ingase ibangele ukungezwani okukhulu komzimba, okuhlanganisa i-angioedema esongela ukuphila. 
  • Izimpawu zingase zihlanganise ukuqubuka, ukulunywa, ukuhoshozela, ukuphefumula kanzima, noma ukuvuvukala kobuso, amehlo, izindebe, ulimi, umphimbo, izandla, imilenze, izinyawo, noma izitho zangasese.
  • Umuthi ungathinta impilo yengqondo, okungase kubangele ukuyaluza, ukucasuka, noma okunye ukuziphatha okungavamile. 
  • I-Pregabalin ingabangela i-edema (ukuvuvukala komzimba) noma ukuzuza kwesisindo, okungase kube yinkinga kubantu abanesifo senhliziyo. 
  • I-Pregabalin ingase futhi yandise ingozi yomdlavuza othile nokopha. Iziguli kufanele zikhulume nodokotela ngezinto ezizikhathazayo.
  • Abesifazane abakhulelwe noma abazama ukukhulelwa kufanele babonane nodokotela wabo ngaphambi kokuthatha i-pregabalin. Abesifazane abancelisayo kufanele bawugweme lo muthi.

Kubalulekile ukuthi ungayeki ukuthatha i-pregabalin kungazelelwe ngaphandle kokubonana nodokotela. Ukuyeka ukuqhubeka kungazelelwe kungase kubangele ukuquleka noma eminye imiphumela emibi ye-pregabalin njengokucasuka, isiyezi, ikhanda elibuhlungu, isicanucanu, ukuhlanza, isifo sohudo, izinkinga zokulala, amaphupho amabi, noma ukuzwa ukuluma.

Isebenza kanjani i-Pregabalin Tablet

I-Pregabalin isebenza ngokubophezela kumasayithi athile ohlelweni lwezinzwa, iguqule ukukhululwa kwe-neurotransmitter, kanye nokuthulisa izinzwa ezisebenza ngokweqile. Le nqubo eyingqayizivele ivumela ukuthi iphathe ngokuphumelelayo izinhlobo ezihlukahlukene zobuhlungu bezinzwa futhi ilawule ukuthunjwa ezigulini zesithuthwane. Ukuguquguquka nokusebenza kwayo kuye kwayenza yaba ithuluzi elibalulekile ekwelapheni izimo zokwelapha eziyinselele eziningana.

Ngingakwazi Ukuthatha I-Pregabalin Ngeminye Imithi?

I-Pregabalin ingasebenzisana nemithi ehlukahlukene nezinto, ikakhulukazi lezo ezinemiphumela emibi efanayo. Okulandelayo kukhona ukuxhumana okuvamile:

  • Ama-Antihistamine, avame ukusetshenziselwa ukungezwani komzimba nezimpawu ezibandayo, angaphinde ahlanganyele ne-pregabalin. 
  • I-Benzodiazepines (BZDs), esetshenziselwa ukwelapha izimo ezifana nokukhathazeka nokuqwasha, ingase ihlanganyele ne-pregabalin, okungase kuholele ekuthungeni ngokweqile kanye nezinkinga zokuphefumula lapho zisetshenziswa ndawonye.
  • I-Glitazones, iqembu lemithi yesifo sikashukela, ingabangela ukunqwabelana koketshezi (i-oedema) uma ihlanganiswa ne-pregabalin. 
  • Ama-opioid, ngokuvamile asetshenziselwa ubuhlungu obukhulu, angasebenzisana kakhulu ne-pregabalin, abangele ukukhathala, isiyezi, nezinkinga zokusebenzisana. 
  • Eminye imithi yokulalisa, ehlanganisa izinsiza zokulala njenge-zolpidem ne-barbiturates, ingasebenzisana ne-pregabalin. 

Ulwazi Lomthamo

Odokotela banquma umthamo ofanele we-pregabalin, ongalungiswa ngokuhamba kwesikhathi ukuze usebenze kahle nokubekezeleleka.

  • Nge-neuropathy yesifo sikashukela, abantu abadala ngokuvamile baqala ngo-50 mg ngomlomo kathathu ngosuku. 
  • Ukwelashwa kwe-postherpetic neuralgia ngokuvamile kuqala ngo-150 kuya ku-300 mg nsuku zonke, kuhlukaniswe imithamo emibili noma emithathu. 
  • Ukuze isithuthwane, umthamo wokuqala ngu-150 mg ngosuku ngemithamo emibili noma emithathu ehlukanisiwe. 
  • Ukwelashwa kwe-Fibromyalgia kuqala ngo-75 mg ngomlomo kabili ngosuku. 
  • Ukwelashwa kobuhlungu be-neuropathic kuqala ku-75 mg ngomlomo kabili ngosuku. 

Isiphetho

I-Pregabalin inomthelela omkhulu ezimpilweni zabantu abaningi ababhekene nobuhlungu bezinzwa, ukukhathazeka, kanye nesifo sokuwa. Ukuguquguquka kwayo ekulawuleni izimo ezihlukahlukene kuyenza ibe ithuluzi elibalulekile kwezokwelapha zesimanje. Kusukela ekudambiseni ubuhlungu be-neuropathic kuya ekulawuleni ukuquleka, ikhono le-pregabalin lokuthulisa izinzwa ezisebenza ngokweqile linikeza induduzo edingeka kakhulu ezigulini ezihlushwa ubuhlungu obungapheli kanye nokuphazamiseka kwemizwa. Nakuba i-pregabalin inikeza izinzuzo eziningi, kubalulekile ukuyisebenzisa njengoba uqondiswa udokotela futhi uqaphele imiphumela yayo engase ibe khona ye-pregabalin nokusebenzisana kwayo. 

FAQ sika

1. Isidakamizwa i-pregabalin sisetshenziselwa ini?

I-Pregabalin isiza ukukhulula ubuhlungu be-neuropathic, obungenzeka ezingalweni, izandla, iminwe, imilenze, izinyawo, noma izinzwane ngenxa yesifo sikashukela noma i-neuralgia ye-postherpetic. Ukwengeza, iphatha i-fibromyalgia kanye nobuhlungu be-neuropathic obubangelwa ukulimala komgogodla. I-Pregabalin iphinde isetshenziswe kanye neminye imithi yokuphatha ukuquleka okuthile kubantu abadala nasezinganeni ezinenyanga eyodwa ubudala nangaphezulu.

2. Ingabe i-pregabalin iphephile ezinso?

Izinso ngokuyinhloko zisusa i-pregabalin. Kubantu abanezinkinga zezinso noma umlando wesifo sezinso, umzimba ungase ungacacisi i-pregabalin ngempumelelo, okungase kuholele ekwenyukeni kwamazinga ezidakamizwa kanye nemiphumela engemihle eyengeziwe. 

3. Yimuphi umphumela ovame kakhulu we-pregabalin?

Imiphumela emibi kakhulu ye-pregabalin yile: 

  • isiyezi 
  • Ukulala
  • Umbono ophundlekile
  • Umlomo omile
  • Inzuzo yesisindo
  • Ukubunzima ukugxila
  • Ukwandisa ukudla

4. Ubani ongakwazi ukuthatha i-pregabalin?

I-Pregabalin ayifanele wonke umuntu. Abantu okufanele bagweme noma basebenzise i-pregabalin ngokuqapha bafaka:

  • Labo abangezwani ne-pregabalin noma izithako zayo
  • Abantu abanezinkinga ezinkulu zezinso
  • Abantu abanomlando wokusebenzisa kabi izidakamizwa noma utshwala
  • abesifazane abakhulelwe noma labo abahlela ukukhulelwa (ngaphandle uma inzuzo engaba khona idlula ingozi)
  • Izingane ezingaphansi kwenyanga eyodwa zokwelashwa kokuquleka

5. Ingabe i-pregabalin iphephile ukuyithatha nsuku zonke?

I-Pregabalin ingathathwa nsuku zonke njengoba kunqunywe udokotela. Kodwa-ke, ukulandela umthamo onqunyiwe we-pregabalin kanye nokubonana nodokotela ngaphambi kokwandisa noma ukwehlisa umthamo kubalulekile. 

6. Kufanele ngithathe isikhathi esingakanani i-pregabalin ukuze ngithole ubuhlungu bezinzwa?

Ubude besikhathi sokwelashwa kwe-pregabalin yobuhlungu bezinzwa siyahlukahluka futhi kuncike ekuphenduleni komuntu ngamunye kanye nesimo sabo esithile. Iziguli akufanele zilindele imiphumela esheshayo, njengoba kungase kuthathe amasonto ambalwa ukuthola izinzuzo ezigcwele ze-pregabalin. 

7. Ingabe i-pregabalin iphephile ukusetshenziswa isikhathi eside?

Nakuba i-pregabalin ingasetshenziswa isikhathi eside ngaphansi kokuqondisa kwezokwelapha, udokotela kufanele ahlole njalo ukuphepha nokusebenza kwayo isikhathi eside. 

8. Ngingakwazi yini ukuthatha i-pregabalin kabili ngosuku?

Yebo, i-pregabalin ingaphuzwa kabili ngosuku, kuye ngomthamo onqunyiwe we-pregabalin kanye nesimo esithile esiphathwayo. Isibonelo, ekwelapheni i-fibromyalgia, umthamo wokuqala uvame ukuba ngu-75 mg kabili ngosuku. 

Umshwana wokuzihlangula: Ulwazi olunikezwe lapha alwenzelwe ukufaka iseluleko esivela kuchwepheshe wezokunakekelwa kwempilo. Ulwazi aluhloselwe ukumboza konke ukusetshenziswa okungenzeka, imiphumela engemihle, izinyathelo zokuphepha, nokusebenzisana kwezidakamizwa. Lolu lwazi aluhloselwe ukuphakamisa ukuthi ukusebenzisa umuthi othile kufanelekile, kuphephile, noma kuyasebenza wena noma omunye umuntu. Ukungabi bikho kwanoma yiluphi ulwazi noma isexwayiso mayelana nomuthi akufanele kuhunyushwe njengesiqinisekiso esicacile esivela enhlanganweni. Sikweluleka ngokuqinile ukuthi uthintane nodokotela uma kukhona okukukhathazayo ngomuthi futhi ungalokothi usebenzise umuthi ngaphandle kwencwadi kadokotela.