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I-Thiocolchicoside

I-Thicolchicoside imithi esetshenziselwa ukukhulula ubuhlungu nokuqina kwemisipha. Ake singene ekuhlaziyeni okuphelele kwe-Thiocolchicoside.

Iyini i-Thiocolchicoside?

I-Thicolchicoside iyi-phytochemical ye-semisynthetic esebenza ngokufana ne-colchicoside yemvelo. Ikhishwa kuma-alkaloid akhiqiza imbewu ezitshalweni. Ngenxa yesenzo saso esivimbela ukuqiniswa kwemisipha, kunciphisa ukuvuvukala, futhi kukhulule ubuhlungu (umbulali wezinhlungu), umuthi wahlukaniswa njengesidakamizwa esiphumuza imisipha, esilwa nokuvuvukala, nesidambisa ubuhlungu. Le ngxenye esebenzayo isebenza ngokushaya ama-receptors athile emzimbeni futhi, ngenxa yalokho, ukwakha ukuvinjelwa kwama-neurotransmitters; kuholela ekunciphiseni imisipha yemisipha, ukuvuvukala, nokuzwela ubuhlungu.

Ukusetshenziswa kwe-Thiocolchicoside

I-Thiocolchicoside imiselwe ngokuyinhloko kubantu abadala abaneminyaka engu-16 noma ngaphezulu ngalezi zimo ezilandelayo:

  • I-Acute noma Engamahlalakhona Ukuhlungu obusemhlane: I-Thiocolchicoside inganciphisa ubuhlungu beqolo ezimweni ezisebenzayo noma ezihlala njalo.
  • Ubuhlungu Bangemva Kokuhlinzwa: Ukuhlinza kungase kucindezele kakhulu, kube nezinsuku eziningi ezibuhlungu. Yilapho inzuzo ye-Thiocolchicoside ilele khona—ikhulula izinhlungu nokugoqeka kwemisipha, okufika kahle ngesikhathi sokululama ngemva kokulimala/ukuhlinzwa.
  • I-Muscle Spasms: Lo muthi unciphisa ukungezwani kwemisipha. Ezinye izinkinga zentamo, ukulimala kwe-arcane, nokulimala kuncishiswa yilo muthi.
  • I-Ankylosing spondylitis (AS) ingenye ye-arthropathies evuthayo evame ukubandakanya umgogodla ekuphathweni okufanele kwezokwelapha. Lokhu kuhlanganisa ukusetshenziswa kwe-Thiocolchicoside njengenye yezidakamizwa.
  • I-rheumatoid Isifo Sokuqaqamba Kwamalunga: Mayelana ne-rheumatoid arthritis, i-Thiocolchicoside ingasiza labo bantu ukuphulukisa imisipha nezinhlungu ezibangelwa yilesi sifo.
  • Ukulimala Komgogodla: Lokhu kulimala engxenyeni yomzimba ezungezile futhi evikela izinzwa, njengomgogodla, kuzokwenza kokubili lesi sidakamizwa kanye ne-Thiocolchicoside kube usizo, njengoba kuzosiza ukugcina ukukhululeka kwemizwa.
  • I-Torticollis Eqhubekayo: Uma i-torticollis ephikisayo (izinto ezisho intamo esontekile entanyeni) iphikelela, sisebenzisa i-Thiocolchicoside, ehlanganisa amaqembu emisipha.

I-Thiocolchicoside Side Effects

I-Thiocolchicoside, njengeminye imithi, ingase ihlotshaniswe nemiphumela ethile engemihle. Eminye yemiphumela emibi evamile ehlobene ne-Thiocolchicoside ihlanganisa:

  • Ukozela noma ukuqunjelwa
  • Ubuhlungu besisu noma ukungakhululeki
  • Gas noma i-flatulence
  • I-nausea
  • Uhudo

Uma ubona noma yimiphi yale miphumela emibi, ehlanganisa ukulunywa, ukuqubuka, ukulahlekelwa ukudla, amehlo abephuzi, ukwehla komfutho wegazi kungazelelwe, noma ukushaya kwenhliziyo okusheshayo, kufanele uqonde egumbini lezokwelapha.

I-Thiocolchicoside Dosage

Uchwepheshe wakho wezokunakekelwa kwempilo kufanele anqume ngomthamo we-Thiocolchicoside ngokucabangela isimo sakho kanye nempumelelo yomuthi esimweni sakho esithile. Nokho, ububanzi bomthamo obujwayelekile bumi kanje:

  • Kubantu abadala: 8 kuya ku-6 mg ngosuku, kuthathwa ngemithamo emi-2 kuye kwemi-3.

Isebenza kanjani i-Thiocolchicoside

I-Thiocolchicoside ishaya isamukeli sesistimu yezinzwa esinciphile esiphethe ukudluliselwa komfutho nokuphumuza imisipha kanye nokuba buthakathaka. Ilingisa ikhemikhali ye-GABA (i-gamma-aminobutyric acid), ehlotshaniswa nethoni yemisipha futhi ivimbe ukuqina. Ngokusebenzisana nalawa ma-receptors, i-Thiocolchicoside ingakwazi:

  • Ukudambisa ubuhlungu obuhlobene nama-muscle spasms nokuqina kwemisipha, kuhlanganise nobuhlungu be-sciatica.
  • Khuthaza ukuphumula kwemisipha

Ukuqapha

Ngaphambi kokuba uqale ukuthatha i-Thiocolchicoside, kufanele wazise udokotela nganoma yiziphi izinkinga zezempilo, izinto ezingezwani nomzimba, nanoma yiziphi ezinye izidakamizwa/imithi oyithathayo. I-Thiocolchicoside kufanele isetshenziswe ngokuqapha noma igwenywe ezimweni ezithile, njenge:

  • ezinzima izinso isifo
  • Umlando wokuquleka
  • Ukungezwani komzimba okuvame kakhulu, njengesifuba somoya noma i-bronchitis.
  • Ukukhulelwa noma ibele.

I-Dose elahlekile

Uma ukhohlwa ukuphuza i-Thiocolchicoside, ungathatha umthamo oqondile uma usukhumbula. Kodwa-ke, uma kuvela ukuthi yisikhathi lapho kufanele ngabe uthathe umthamo olandelayo, vele uyeke ukuthatha umthamo ogejiwe futhi ugcine uhlelo olujwayelekile. Gwema ukuphinda umthamo ukuze uwuthathe futhi, ngoba kungenza inqubo yokwelapha ibe nzima.

ukweqisa izidakamizwa

Esimeni sokudlula umthamo noma okusolakala ukuthi ukweqisa kwe-Thiocolchicoside, ukufuna iseluleko sikadokotela kubalulekile, noma ukushayela isikhungo sokulawula ubuthi. Izimpawu zokweqisa zingase zihlanganise ubuthongo obungavamile, ukungakwazi ukuhlonza isiqondiso esifanele okwesikhashana noma ukuhlupheka. ukuphelelwa umoya.

I-Thiocolchicoside Storage

Gcina i-Thiocolchicoside ekamelweni lokushisa ukuze ingavezwa umswakama nokukhanya kwelanga. Khumbula ukuthi izingane nezilwane ezifuywayo zingase ziwuthole ngephutha umuthi. Ukuvimbela lokhu, beka imithi eduze ngangokunokwenzeka lapho ingakwazi ukufinyelela khona. Gwema ukusebenzisa ukwelashwa kwe-Thiocolchicoside lapho idethi yokuphelelwa yisikhathi isiphelile noma ngemva kwesikhathi esinqunyiwe.

Ukuqhathanisa: Thiocolchicoside vs Chlorzoxazone

Kokubili i-Thiocolchicoside ne-chlorzoxazone iziphumuli zemisipha ezisetshenziselwa ukwelapha ukugogeka kwemisipha. Nakuba zinemiphumela efanayo yokwelapha, kunomehluko othile:

Point

I-Thiocolchicoside

I-Chlorzoxazone

I-Drug Class

Ukuphumuza imisipha

Ukuphumuza imisipha

Indlela Yokusebenza

Isebenza kuma-GABA receptors ohlelweni lwezinzwa ukunciphisa ukuqina kwemisipha nokuqina

Isebenza phakathi nendawo ukuze icindezele umsebenzi wama-motor neurons kuntambo yomgogodla kanye ne-brainstem

Izinkomba

Isetshenziselwa ukwelapha ama-musculoskeletal spasms, ukuqina, nobuhlungu obuhambisana nezimo ezihlukahlukene ze-musculoskeletal

Isetshenziselwa ukwelapha ama-musculoskeletal spasms, ubuhlungu, nokungakhululeki okuhambisana nezimo ezibuhlungu nezibuhlungu ze-musculoskeletal.

 Izakhiwo ezingeziwe

I-anti-inflammatory kanye ne-analgesic (eqeda ubuhlungu).

Akukho okushiwo ngokuqondile ngezakhiwo ezengeziwe zokulwa nokuvuvukala noma zokuqeda ukuvuvukala

Imiphumela Ejwayelekile Ejwayelekile

Ukozela, ubuhlungu besisu, isicanucanu, isifo sohudo

Ukozela, isiyezi, isicanucanu, ukuhlanza

Isiphetho

I-Thiocolchicoside umuthi osebenzayo ongadambisa imisipha, ukuqina, nobuhlungu obuhambisana nezimo ezahlukahlukene ze-musculoskeletal. Iqondise ama-receptors athile ohlelweni lwezinzwa, ikhuthaza ukuphumula kwemisipha nokunciphisa ukuvuvukala. Kodwa-ke, kubalulekile ukusebenzisa i-Thiocolchicoside ngaphansi kokuqondisa kochwepheshe bezempilo futhi ulandele umthamo onqunyiwe kanye nezinyathelo zokuphepha ukuze unciphise ubungozi bemiphumela emibi. Ngokusetshenziswa kahle, i-Thiocolchicoside ingaba inketho yokwelapha ephumelelayo yokuphatha izindaba eziphathelene nemisipha kanye nokwenza ngcono ikhwalithi yokuphila iyonke.

FAQ sika

1. Ingabe i-Thiocolchicoside iphephile? 

I-Thiocolchicoside ngokuvamile iphephile uma ithathwa njengoba kuyalelwe uchwepheshe wezokunakekelwa kwempilo. Kodwa-ke, njenganoma yimuphi umuthi, ungabangela imiphumela emibi, futhi kufanele kulandelwe izinyathelo ezithile zokuphepha. Kubalulekile ukuxoxa ngomlando wakho wezokwelapha nanoma yiziphi izingozi ezingase zibe khona nodokotela wakho ngaphambi kokuthatha i-Thiocolchicoside.

2. Ingabe i-Thiocolchicoside iyiphilisi lezinhlungu? 

Nakuba i-Thiocolchicoside ingesona isidambisi sezinhlungu ngokuyinhloko, inezindawo zokudambisa izinhlungu (ezidambisa izinhlungu) ngenxa yemiphumela yayo eqeda ukuvuvukala. Kodwa-ke, isetshenziswa ngokuyinhloko njenge-relax ye-muscle ekwelapheni ama-muscle spasms nokuqina.

3. Ingabe i-Thiocolchicoside iyi-steroid? 

Cha, i-Thiocolchicoside ayiyona i-steroid. Iphuma ku-semisynthetic ye-colchicoside eyakhiwe ngokwemvelo, etholakala embewini yesitshalo i-Gloriosa superba, evame ukubizwa ngokuthi i-flame lily noma i-global lily.

4. Yikuphi okungcono: I-Chlorzoxazone noma i-Thiocolchicoside? 

Kokubili i-Thiocolchicoside ne-chlorzoxazone iziphumuli zemisipha ezisebenzayo ezisetshenziselwa ukwelapha ukugogeka kwemisipha. Nakuba ezinye izifundo zibonise ukuthi i-chlorzoxazone isebenza kancane, umehluko udinga ubaluleke kakhulu ukuze ube nenjongo yomtholampilo. Umhlinzeki wakho wokunakekelwa kwezempilo uzonquma inketho efanelekile kakhulu ngokusekelwe esimweni sakho esithile kanye nezidingo zomuntu ngamunye.

5. Ungathatha isikhathi esingakanani i-Thiocolchicoside? 

Ubude besikhathi sokwelashwa kwe-Thiocolchicoside buncike ebukhulwini besimo sakho futhi kufanele bunqunywe umhlinzeki wakho wokunakekelwa kwezempilo. Ukulandela umthamo onqunyiwe futhi ungadluli isikhathi esinconywayo kubalulekile ngaphandle kokubonisana nodokotela wakho.

6. Ingabe i-Thiocolchicoside iphephile phakathi ukukhulelwa

I-Thiocolchicoside ayinconywa ukuthi isetshenziswe ngesikhathi sokukhulelwa noma ukuncelisa, njengoba ingase ibe nemiphumela emibi ku-fetus ekhulayo noma usana oluncelisayo. Kubalulekile ukwazisa umhlinzeki wakho wezempilo uma ukhulelwe, uhlela ukukhulelwa, noma uncelisa ngaphambi kokuthatha i-Thiocolchicoside.

7. Ingabe i-Thiocolchicoside iyalutha? 

Cha, i-Thiocolchicoside ayithathwa njengomuthi oluthayo. Kodwa-ke, kusabalulekile ukulandela umthamo onqunyiwe kanye nemiyalelo ehlinzekwa nguchwepheshe wakho wezempilo ukuze ugweme noma yiziphi izingozi ezingaba khona noma imiphumela emibi.