I-Thicolchicoside imithi esetshenziselwa ukukhulula ubuhlungu nokuqina kwemisipha. Ake singene ekuhlaziyeni okuphelele kwe-Thiocolchicoside.
I-Thicolchicoside iyi-phytochemical ye-semisynthetic esebenza ngokufana ne-colchicoside yemvelo. Ikhishwa kuma-alkaloid akhiqiza imbewu ezitshalweni. Ngenxa yesenzo saso esivimbela ukuqiniswa kwemisipha, kunciphisa ukuvuvukala, futhi kukhulule ubuhlungu (umbulali wezinhlungu), umuthi wahlukaniswa njengesidakamizwa esiphumuza imisipha, esilwa nokuvuvukala, nesidambisa ubuhlungu. Le ngxenye esebenzayo isebenza ngokushaya ama-receptors athile emzimbeni futhi, ngenxa yalokho, ukwakha ukuvinjelwa kwama-neurotransmitters; kuholela ekunciphiseni imisipha yemisipha, ukuvuvukala, nokuzwela ubuhlungu.
I-Thiocolchicoside imiselwe ngokuyinhloko kubantu abadala abaneminyaka engu-16 noma ngaphezulu ngalezi zimo ezilandelayo:
I-Thiocolchicoside, njengeminye imithi, ingase ihlotshaniswe nemiphumela ethile engemihle. Eminye yemiphumela emibi evamile ehlobene ne-Thiocolchicoside ihlanganisa:
Uma ubona noma yimiphi yale miphumela emibi, ehlanganisa ukulunywa, ukuqubuka, ukulahlekelwa ukudla, amehlo abephuzi, ukwehla komfutho wegazi kungazelelwe, noma ukushaya kwenhliziyo okusheshayo, kufanele uqonde egumbini lezokwelapha.
Uchwepheshe wakho wezokunakekelwa kwempilo kufanele anqume ngomthamo we-Thiocolchicoside ngokucabangela isimo sakho kanye nempumelelo yomuthi esimweni sakho esithile. Nokho, ububanzi bomthamo obujwayelekile bumi kanje:
I-Thiocolchicoside ishaya isamukeli sesistimu yezinzwa esinciphile esiphethe ukudluliselwa komfutho nokuphumuza imisipha kanye nokuba buthakathaka. Ilingisa ikhemikhali ye-GABA (i-gamma-aminobutyric acid), ehlotshaniswa nethoni yemisipha futhi ivimbe ukuqina. Ngokusebenzisana nalawa ma-receptors, i-Thiocolchicoside ingakwazi:
Ngaphambi kokuba uqale ukuthatha i-Thiocolchicoside, kufanele wazise udokotela nganoma yiziphi izinkinga zezempilo, izinto ezingezwani nomzimba, nanoma yiziphi ezinye izidakamizwa/imithi oyithathayo. I-Thiocolchicoside kufanele isetshenziswe ngokuqapha noma igwenywe ezimweni ezithile, njenge:
Uma ukhohlwa ukuphuza i-Thiocolchicoside, ungathatha umthamo oqondile uma usukhumbula. Kodwa-ke, uma kuvela ukuthi yisikhathi lapho kufanele ngabe uthathe umthamo olandelayo, vele uyeke ukuthatha umthamo ogejiwe futhi ugcine uhlelo olujwayelekile. Gwema ukuphinda umthamo ukuze uwuthathe futhi, ngoba kungenza inqubo yokwelapha ibe nzima.
Esimeni sokudlula umthamo noma okusolakala ukuthi ukweqisa kwe-Thiocolchicoside, ukufuna iseluleko sikadokotela kubalulekile, noma ukushayela isikhungo sokulawula ubuthi. Izimpawu zokweqisa zingase zihlanganise ubuthongo obungavamile, ukungakwazi ukuhlonza isiqondiso esifanele okwesikhashana noma ukuhlupheka. ukuphelelwa umoya.
Gcina i-Thiocolchicoside ekamelweni lokushisa ukuze ingavezwa umswakama nokukhanya kwelanga. Khumbula ukuthi izingane nezilwane ezifuywayo zingase ziwuthole ngephutha umuthi. Ukuvimbela lokhu, beka imithi eduze ngangokunokwenzeka lapho ingakwazi ukufinyelela khona. Gwema ukusebenzisa ukwelashwa kwe-Thiocolchicoside lapho idethi yokuphelelwa yisikhathi isiphelile noma ngemva kwesikhathi esinqunyiwe.
Kokubili i-Thiocolchicoside ne-chlorzoxazone iziphumuli zemisipha ezisetshenziselwa ukwelapha ukugogeka kwemisipha. Nakuba zinemiphumela efanayo yokwelapha, kunomehluko othile:
|
Point |
I-Thiocolchicoside |
I-Chlorzoxazone |
|
I-Drug Class |
Ukuphumuza imisipha |
Ukuphumuza imisipha |
|
Indlela Yokusebenza |
Isebenza kuma-GABA receptors ohlelweni lwezinzwa ukunciphisa ukuqina kwemisipha nokuqina |
Isebenza phakathi nendawo ukuze icindezele umsebenzi wama-motor neurons kuntambo yomgogodla kanye ne-brainstem |
|
Izinkomba |
Isetshenziselwa ukwelapha ama-musculoskeletal spasms, ukuqina, nobuhlungu obuhambisana nezimo ezihlukahlukene ze-musculoskeletal |
Isetshenziselwa ukwelapha ama-musculoskeletal spasms, ubuhlungu, nokungakhululeki okuhambisana nezimo ezibuhlungu nezibuhlungu ze-musculoskeletal. |
|
Izakhiwo ezingeziwe |
I-anti-inflammatory kanye ne-analgesic (eqeda ubuhlungu). |
Akukho okushiwo ngokuqondile ngezakhiwo ezengeziwe zokulwa nokuvuvukala noma zokuqeda ukuvuvukala |
|
Imiphumela Ejwayelekile Ejwayelekile |
Ukozela, ubuhlungu besisu, isicanucanu, isifo sohudo |
Ukozela, isiyezi, isicanucanu, ukuhlanza |
I-Thiocolchicoside umuthi osebenzayo ongadambisa imisipha, ukuqina, nobuhlungu obuhambisana nezimo ezahlukahlukene ze-musculoskeletal. Iqondise ama-receptors athile ohlelweni lwezinzwa, ikhuthaza ukuphumula kwemisipha nokunciphisa ukuvuvukala. Kodwa-ke, kubalulekile ukusebenzisa i-Thiocolchicoside ngaphansi kokuqondisa kochwepheshe bezempilo futhi ulandele umthamo onqunyiwe kanye nezinyathelo zokuphepha ukuze unciphise ubungozi bemiphumela emibi. Ngokusetshenziswa kahle, i-Thiocolchicoside ingaba inketho yokwelapha ephumelelayo yokuphatha izindaba eziphathelene nemisipha kanye nokwenza ngcono ikhwalithi yokuphila iyonke.
I-Thiocolchicoside ngokuvamile iphephile uma ithathwa njengoba kuyalelwe uchwepheshe wezokunakekelwa kwempilo. Kodwa-ke, njenganoma yimuphi umuthi, ungabangela imiphumela emibi, futhi kufanele kulandelwe izinyathelo ezithile zokuphepha. Kubalulekile ukuxoxa ngomlando wakho wezokwelapha nanoma yiziphi izingozi ezingase zibe khona nodokotela wakho ngaphambi kokuthatha i-Thiocolchicoside.
Nakuba i-Thiocolchicoside ingesona isidambisi sezinhlungu ngokuyinhloko, inezindawo zokudambisa izinhlungu (ezidambisa izinhlungu) ngenxa yemiphumela yayo eqeda ukuvuvukala. Kodwa-ke, isetshenziswa ngokuyinhloko njenge-relax ye-muscle ekwelapheni ama-muscle spasms nokuqina.
Cha, i-Thiocolchicoside ayiyona i-steroid. Iphuma ku-semisynthetic ye-colchicoside eyakhiwe ngokwemvelo, etholakala embewini yesitshalo i-Gloriosa superba, evame ukubizwa ngokuthi i-flame lily noma i-global lily.
Kokubili i-Thiocolchicoside ne-chlorzoxazone iziphumuli zemisipha ezisebenzayo ezisetshenziselwa ukwelapha ukugogeka kwemisipha. Nakuba ezinye izifundo zibonise ukuthi i-chlorzoxazone isebenza kancane, umehluko udinga ubaluleke kakhulu ukuze ube nenjongo yomtholampilo. Umhlinzeki wakho wokunakekelwa kwezempilo uzonquma inketho efanelekile kakhulu ngokusekelwe esimweni sakho esithile kanye nezidingo zomuntu ngamunye.
Ubude besikhathi sokwelashwa kwe-Thiocolchicoside buncike ebukhulwini besimo sakho futhi kufanele bunqunywe umhlinzeki wakho wokunakekelwa kwezempilo. Ukulandela umthamo onqunyiwe futhi ungadluli isikhathi esinconywayo kubalulekile ngaphandle kokubonisana nodokotela wakho.
I-Thiocolchicoside ayinconywa ukuthi isetshenziswe ngesikhathi sokukhulelwa noma ukuncelisa, njengoba ingase ibe nemiphumela emibi ku-fetus ekhulayo noma usana oluncelisayo. Kubalulekile ukwazisa umhlinzeki wakho wezempilo uma ukhulelwe, uhlela ukukhulelwa, noma uncelisa ngaphambi kokuthatha i-Thiocolchicoside.
Cha, i-Thiocolchicoside ayithathwa njengomuthi oluthayo. Kodwa-ke, kusabalulekile ukulandela umthamo onqunyiwe kanye nemiyalelo ehlinzekwa nguchwepheshe wakho wezempilo ukuze ugweme noma yiziphi izingozi ezingaba khona noma imiphumela emibi.